Discovery of pyrazine carboxamide CB1 antagonists: The introduction of a hydroxyl group improves the pharmaceutical properties and in vivo efficacy of the series-Reference-Cited by-同舟云学术

Discovery of pyrazine carboxamide CB1 antagonists: The introduction of a hydroxyl group improves the pharmaceutical properties and in vivo efficacy of the series

Published:2007-07 Issue:14 Volume:17 Page:3978-3982
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Ellsworth Bruce A.,Wang Ying,Zhu Yeheng,Pendri Annapurna,Gerritz Samuel W.,Sun Chongqing,Carlson Kenneth E.,Kang Liya,Baska Rose A.,Yang Yifan,Huang Qi,Burford Neil T.,Cullen Mary Jane,Johnghar Susan,Behnia Kamelia,Pelleymounter Mary Ann,Washburn William N.,Ewing William R.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference31 articles.

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4. A Potential Decline in Life Expectancy in the United States in the 21st Century

5. The Emerging Role of the Endocannabinoid System in Endocrine Regulation and Energy Balance

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