Optimisation of momelotinib with improved potency and efficacy as pan-JAK inhibitor-Reference-Cited by-同舟云学术

Optimisation of momelotinib with improved potency and efficacy as pan-JAK inhibitor

Published:2022-06 Issue: Volume:66 Page:128728
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Desai Jigar,Patel Bhaumin,Gite Archana,Panchal Nandini,Gite Sanjay,Argade Anil,Kumar Jeevan,Sachchidanand S.,Bandyopadhyay Debdutta,Ghoshdastidar Krishnarup,Patel Hoshang,Chatterjee Abhijit,Mahapatra Jogeshwar,Sharma Manoranjan,Giri Poonam,Kumar Sanjay,Jain Mukul,Sharma Rajiv,Desai Ranjit

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference20 articles.

1. Inborn errors of human JAKs and STATs;Casanova;Immunity.,2012

2. Cytokine receptor signaling through the Jak-Stat-Socs pathway in disease;O'Sullivan;Mol Immunol.,2007

3. Janus kinases in immune cell signaling;Kamran;Immunol Rev.,2009

4. Intracellular signal pathways: potential for therapies;Mavers;Curr Rheumatol Rep.,2009

5. The Janus Kinases (JAKs);Yamaoka;Genome Biol.,2004

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