Discovery and characterization of potent and selective 4-oxo-4-(5-(5-phenyl-1,2,4-oxadiazol-3-yl)indolin-1-yl)butanoic acids as S1P1 agonists-Reference-Cited by-同舟云学术

Discovery and characterization of potent and selective 4-oxo-4-(5-(5-phenyl-1,2,4-oxadiazol-3-yl)indolin-1-yl)butanoic acids as S1P1 agonists

Published:2011-10 Issue:19 Volume:21 Page:6013-6018
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Buzard Daniel,Han Sangdon,Thoresen Lars,Moody Jeanne,Lopez Luis,Kawasaki Andrew,Schrader Thomas,Sage Carleton,Gao Yinghong,Edwards Jeff,Barden Jeremy,Thatte Jayant,Fu Lixia,Solomon Michelle,Liu Ling,Al-Shamma Hussien,Gatlin Joel,Le Minh,Xing Charles,Espinola Sheryll,Jones Robert M.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference11 articles.

1. FTY720 (fingolimod) in Multiple Sclerosis: therapeutic effects in the immune and the central nervous system

2. Sphingosine-1-phosphate and immune regulation: trafficking and beyond

3. Chapter 16 Sphingosine 1-Phosphate Type 1 Receptor Modulators: Recent Advances and Therapeutic Potential

4. .

5. Effect of FTY720, a novel immunosuppressant, on adjuvant-induced arthritis in rats

Cited by 10 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Modulators of Sphingosine-1-phosphate Pathway Biology: Recent Advances of Sphingosine-1-phosphate Receptor 1 (S1P1) Agonists and Future Perspectives;Journal of Medicinal Chemistry;2017-03-30

2. Continuous-flow synthesis of highly functionalized imidazo-oxadiazoles facilitated by microfluidic extraction;Beilstein Journal of Organic Chemistry;2017-02-07

3. Identification of 3,5,6-substituted indolin-2-one’s inhibitors of Aurora B by development of a luminescent kinase assay;Bioorganic & Medicinal Chemistry Letters;2015-08

4. Discovery of APD334: Design of a Clinical Stage Functional Antagonist of the Sphingosine-1-phosphate-1 Receptor;ACS Medicinal Chemistry Letters;2014-11-04

5. Novel S1P1 Receptor Agonists − Part 3: From Thiophenes to Pyridines;Journal of Medicinal Chemistry;2013-12-24