Conversion of 4-cyanomethyl-pyrazole-3-carboxamides into CB1 antagonists with lowered propensity to pass the blood–brain-barrier-Reference-Cited by-同舟云学术

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Conversion of 4-cyanomethyl-pyrazole-3-carboxamides into CB1 antagonists with lowered propensity to pass the blood–brain-barrier

Published:2010-01 Issue:2 Volume:20 Page:453-457
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Receveur Jean-Marie,Murray Anthony,Linget Jean-Michel,Nørregaard Pia K.,Cooper Martin,Bjurling Emelie,Nielsen Peter Aadal,Högberg Thomas

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference28 articles.

1. The endocannabinoid system: Its general strategy of action, tools for its pharmacological manipulation and potential therapeutic exploitation

2. An introduction to the endocannabinoid system: from the early to the latest concepts

3. The endocannabinoid system as a link between homoeostatic and hedonic pathways involved in energy balance regulation

4. Cannabinoid receptor antagonists: pharmacological opportunities, clinical experience, and translational prognosis

5. CB1 receptor antagonism: biological basis for metabolic effects

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1. Optimizing and characterizing 4-methyl substituted pyrazol-3-carboxamides leading to the peripheral cannabinoid 1 receptor inverse agonist TM38837;Bioorganic & Medicinal Chemistry Letters;2024-01

2. Liquid extraction surface analysis‐mass spectrometry: An advanced and environment‐friendly analytical tool in modern analysis;Journal of Separation Science;2022-05-23

3. Anti-obesity therapy with peripheral CB1 blockers: from promise to safe(?) practice;International Journal of Obesity;2020-04-21

4. The therapeutic potential of second and third generation CB1R antagonists;Pharmacology & Therapeutics;2020-04

5. Cannabis: From a Plant That Modulates Feeding Behaviors toward Developing Selective Inhibitors of the Peripheral Endocannabinoid System for the Treatment of Obesity and Metabolic Syndrome;Toxins;2019-05-15

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