3-Indolyl sultams as selective CRTh2 antagonists-Reference-Cited by-同舟云学术

3-Indolyl sultams as selective CRTh2 antagonists

Published:2010-06 Issue:11 Volume:20 Page:3287-3290
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Tumey L. Nathan,Robarge Michael J.,Gleason Elizabeth,Song Jianping,Murphy Steven M.,Ekema George,Doucette Chris,Hanniford Doug,Palmer Marc,Pawlowski Gary,Danzig Joel,Loftus Margaret,Hunady Karen,Sherf Bruce,Mays Robert W.,Stricker-Krongrad Alain,Brunden Kurt R.,Bennani Youssef L.,Harrington John J.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference21 articles.

1. Evidence for Elevated Levels of Histamine, Prostaglandin D2, and Other Bronchoconstricting Prostaglandins in the Airways of Subjects with Mild Asthma

2. Prostanoid Receptors: Structures, Properties, and Functions

3. Chemoattractant Receptors Expressed on Type 2 T Cells and Their Role in Disease

4. CRTH2, an orphan receptor of T-helper-2-cells, is expressed on basophils and eosinophils and responds to mast cell-derived factor(s)

5. Prostaglandin D2 Selectively Induces Chemotaxis in T Helper Type 2 Cells, Eosinophils, and Basophils via Seven-Transmembrane Receptor Crth2

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