Discovery of 7-azaindole derivatives as potent Orai inhibitors showing efficacy in a preclinical model of asthma-Reference-Cited by-同舟云学术

Discovery of 7-azaindole derivatives as potent Orai inhibitors showing efficacy in a preclinical model of asthma

Published:2015-03 Issue:6 Volume:25 Page:1217-1222
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Esteve Cristina,González Jacob,Gual Sílvia,Vidal Laura,Alzina Soledad,Sentellas Sonia,Jover Irene,Horrillo Raquel,De Alba Jorge,Miralpeix Montserrat,Tarrasón Gema,Vidal Bernat

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference14 articles.

1. Physiological and pathophysiological functions of SOCE in the immune system

2. Calcium signaling in the development and function of T-lineage cells

3. CRACM1 Is a Plasma Membrane Protein Essential for Store-Operated Ca 2+ Entry

4. Defective mast cell effector functions in mice lacking the CRACM1 pore subunit of store-operated calcium release–activated calcium channels

5. Store-operated CRAC channels: function in health and disease

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