Low entropic cost of binding confers high selectivity on an allosteric ERK2 inhibitor
Author:
Funder
Osaka Metropolitan University
Publisher
Elsevier BV
Subject
Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry
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1. Distinct binding modes of a benzothiazole derivative confer structural bases for increasing ERK2 or p38α MAPK selectivity;Biochemical and Biophysical Research Communications;2024-04
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