Rational design, synthesis and structure–activity relationships of a cyclic succinate series of TNF-α converting enzyme inhibitors. Part 2: lead optimization-Reference-Cited by-同舟云学术

Rational design, synthesis and structure–activity relationships of a cyclic succinate series of TNF-α converting enzyme inhibitors. Part 2: lead optimization

Published:2003-12 Issue:24 Volume:13 Page:4299-4304
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Xue Chu-Biao,He Xiaohua,Roderick John,Corbett Ronald L,Duan James J.-W,Liu Rui-Qin,Covington Maryanne B,Qian Mingxin,Ribadeneira Maria D,Vaddi Krishna,Christ David D,Newton Robert C,Trzaskos James M,Magolda Ronald L,Wexler Ruth R,Decicco Carl P

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference28 articles.

1. Human tumor necrosis factor. Production, purification, and characterization.

2. Taming TNF: strategies to restrain this proinflammatory cytokine

3. Therapeutic Potential and Strategies for Inhibiting Tumor Necrosis Factor-α

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