Bioisosteric replacement of dihydropyrazole of 4S-(−)-3-(4-chlorophenyl)-N-methyl-N′-[(4-chlorophenyl)-sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-caboxamidine (SLV-319) a potent CB1 receptor antagonist by imidazole and oxazole-Reference-Cited by-同舟云学术

Bioisosteric replacement of dihydropyrazole of 4S-(−)-3-(4-chlorophenyl)-N-methyl-N′-[(4-chlorophenyl)-sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-caboxamidine (SLV-319) a potent CB1 receptor antagonist by imidazole and oxazole

Published:2008-02 Issue:3 Volume:18 Page:963-968
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Srivastava Brijesh Kumar,Soni Rina,Joharapurkar Amit,Sairam Kalapatapu V.V.M.,Patel Jayendra Z.,Goswami Amitgiri,Shedage Sandeep A.,Kar Sidhartha S.,Salunke Rahul P.,Gugale Shivaji B.,Dhawas Amol,Kadam Pravin,Mishra Bhupendra,Sadhwani Nisha,Unadkat Vishal B.,Mitra Prasenjit,Jain Mukul R.,Patel Pankaj R.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

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