Discovery of a spiroindane based compound as a potent, selective, orally bioavailable melanocortin subtype-4 receptor agonist-Reference-Cited by-同舟云学术

Discovery of a spiroindane based compound as a potent, selective, orally bioavailable melanocortin subtype-4 receptor agonist

Published:2010-04 Issue:7 Volume:20 Page:2106-2110
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

He Shuwen,Ye Zhixiong,Dobbelaar Peter H.,Sebhat Iyassu K.,Guo Liangqin,Liu Jian,Jian Tianying,Lai Yingjie,Franklin Christopher L.,Bakshi Raman K.,Dellureficio James P.,Hong Qingmei,Tsou Nancy N.,Ball Richard G.,Cashen Doreen E.,Martin William J.,Weinberg David H.,MacNeil Tanya,Tang Rui,Tamvakopoulos Constantin,Peng Qianping,Miller Randy R.,Stearns Ralph A.,Chen Howard Y.,Chen Airu S.,Strack Alison M.,Fong Tung M.,MacIntyre D. Euan,Wyvratt Matthew J.,Nargund Ravi P.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference45 articles.

1. Studies on the Physiological Functions of the Melanocortin System

2. The melanocortin system

3. Recent developments in our understanding of melanocortin system in the regulation of food intake

4. Anatomy and regulation of the central melanocortin system

5. Divergence of Melanocortin Pathways in the Control of Food Intake and Energy Expenditure

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