Design and synthesis of selective keto-1,2,4-oxadiazole-based tryptase inhibitors-Reference-Cited by-同舟云学术

Design and synthesis of selective keto-1,2,4-oxadiazole-based tryptase inhibitors

Published:2006-07 Issue:13 Volume:16 Page:3434-3439
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Palmer James T.,Rydzewski Robert M.,Mendonca Rohan V.,Sperandio David,Spencer Jeffrey R.,Hirschbein Bernard L.,Lohman Julia,Beltman Jeri,Nguyen Margaret,Liu Liang

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference16 articles.

1. Inhibitors of mast cell tryptase beta as therapeutics for the treatment of asthma and inflammatory disorders

2. Mast cell tryptase: a review of its physiology and clinical significance

3. Mast cell tryptase, a still enigmatic enzyme

4. Caughey, G. H. Handbook of Proteolytic Enzymes, 2nd ed., 2004; Vol. 2, p 1535.

5. The role of the mast cell in asthma: a reassessment

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