Synthesis and structure–activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 2-Reference-Cited by-同舟云学术

Synthesis and structure–activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 2

Published:2006-09 Issue:18 Volume:16 Page:4922-4930
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Hudson Sarah,Kiankarimi Mehrak,Rowbottom Martin W.,Vickers Troy D.,Wu Dongpei,Pontillo Joseph,Ching Brett,Dwight Wesley,Goodfellow Val S.,Schwarz David,Heise Christopher E.,Madan Ajay,Wen Jenny,Ban William,Wang Hua,Wade Warren S.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference31 articles.

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2. Melanin-concentrating hormone and its receptors: state of the art

3. Binding sites for melanin-concentrating hormone in the human brain

4. T-226296: a novel, orally active and selective melanin-concentrating hormone receptor antagonist

5. Erratum: Antidepressant, anxiolytic and anorectic effects of a melanin-concentrating hormone-1 receptor antagonist

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