Discovery of a novel 2-(1 H -pyrazolo[3,4- b ]pyridin-1-yl)thiazole derivative as an EP 1 receptor antagonist and in vivo studies in a bone fracture model
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry
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1. Prostanoids in health and disease
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3. Prostaglandin facilitates afferent nerve activity via EP1 receptors during urinary bladder inflammation in rats
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5. Hit-to-lead optimization of 2-(1H-pyrazol-1-yl)-thiazole derivatives as a novel class of EP1 receptor antagonists
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1. Discovery of New 1,4,6-Trisubstituted-1H-pyrazolo[3,4-b]pyridines with Anti-Tumor Efficacy in Mouse Model of Breast Cancer;Pharmaceutics;2023-02-27
2. One-pot three-component synthesis of novel pyrazolo[3,4-b]pyridines as potent antileukemic agents;European Journal of Medicinal Chemistry;2022-01
3. Diverse N-Substituted Azole-Containing Amino Acids as Building Blocks for Cyclopeptides;ACS Omega;2020-01-08
4. Adjuvant drug-assisted bone healing: Part I – Modulation of inflammation;Clinical Hemorheology and Microcirculation;2020-01-03
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