N1-arylsulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole derivatives are potent and selective 5-HT6 receptor antagonists-Reference-Cited by-同舟云学术

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N1-arylsulfonyl-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole derivatives are potent and selective 5-HT6 receptor antagonists

Published:2005-01 Issue:2 Volume:15 Page:379-383
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Cole Derek C.,Ellingboe John W.,Lennox William J.,Mazandarani Hossein,Smith Deborah L.,Stock Joseph R.,Zhang Guoming,Zhou Ping,Schechter Lee E.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference19 articles.

1. A Novel Rat Serotonin (5-HT6) Receptor: Molecular Cloning, Localization and Stimulation of cAMP Accumulation

2. Cloning, Characterization, and Chromosomal Localization of a Human 5-HT6 Serotonin Receptor

3. 5-HT6 receptors positively coupled to adenylyl cyclase in striatal neurones in culture

4. 5-ht6 Receptors

Cited by 42 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Copper-catalyzed N-arylation of pyrroles: an overview;New Journal of Chemistry;2021

2. 2-Aminoimidazole-based antagonists of the 5-HT6 receptor – A new concept in aminergic GPCR ligand design;European Journal of Medicinal Chemistry;2019-10

3. Synthesis, Structural and Thermal Studies of 3-(1-Benzyl-1,2,3,6-tetrahydropyridin-4-yl)-5-ethoxy-1H-indole (D2AAK1_3) as Dopamine D2 Receptor Ligand;Molecules;2018-09-04

4. Discovery and Development of 1-[(2-Bromophenyl)sulfonyl]-5-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dimesylate Monohydrate (SUVN-502): A Novel, Potent, Selective and Orally Active Serotonin 6 (5-HT6) Receptor Antagonist for Potential Treatment of Alzheimer’s Disease;Journal of Medicinal Chemistry;2017-02-17

5. Synthesis and biological evaluation of novel N1-phenylsulphonyl indole derivatives as potent and selective 5-HT6R ligands for the treatment of cognitive disorders;Journal of Enzyme Inhibition and Medicinal Chemistry;2016-11-01

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