Synthesis and preliminary evaluation of 4-hydroxy-6-(3-[11C]methoxyphenethyl)pyridazin-3(2H)-one, a 11C-labeled -amino acid oxidase (DAAO) inhibitor for PET imaging-Reference-Cited by-同舟云学术

Synthesis and preliminary evaluation of 4-hydroxy-6-(3-[11C]methoxyphenethyl)pyridazin-3(2H)-one, a 11C-labeled -amino acid oxidase (DAAO) inhibitor for PET imaging

Published:2020-08 Issue:16 Volume:30 Page:127326
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Deng Xiaoyun,Zhang Yiding,Chen Zhen,Kumata Katsushi,Van Richard,Rong Jian,Shao Tuo,Hatori Akiko,Mori Wakana,Yu Qingzhen,Hu Kuan^ORCID,Fujinaga Masayuki,Wey Hsiao-Ying,Shao Yihan,Josephson Lee,Murtas Giulia,Pollegioni Loredano,Zhang Ming-Rong,Liang Steven^ORCID

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

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4. D-amino acid oxidase gene therapy sensitizes glioma cells to the antiglycolytic effect of 3-bromopyruvate

5. Enzymatic assay of d-serine using d-serine dehydratase from Saccharomyces cerevisiae

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