Discovery of (3S,4S)-3-methyl-3-(4-fluorophenyl)-4-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxyprop-2-yl)phenyl)pyrrolidines as novel RORγt inverse agonists-Reference-Cited by-同舟云学术

Discovery of (3S,4S)-3-methyl-3-(4-fluorophenyl)-4-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxyprop-2-yl)phenyl)pyrrolidines as novel RORγt inverse agonists

Published:2020-09 Issue:17 Volume:30 Page:127392
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Jiang Bin^ORCID,Duan James J.-W.^ORCID,Stachura Sylwia,Karmakar Ananta,Hemagiri Hemalatha,Raut Dhanya Kumar,Gupta Arun Kumar,Weigelt Carolyn A.,Khan Javed,Sack John S.,Wu Dauh-Rurng,Yarde Melissa,Shen Ding-Ren,Galella Michael A.,Mathur Arvind,Zhao Qihong,Salter-Cid Luisa M.,Carter Percy H.,Dhar T.G. Murali

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference19 articles.

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