Challenges in the development of an M 4 PAM preclinical candidate: The discovery, SAR, and biological characterization of a series of azetidine-derived tertiary amides-Reference-Cited by-同舟云学术

Challenges in the development of an M 4 PAM preclinical candidate: The discovery, SAR, and biological characterization of a series of azetidine-derived tertiary amides

Published:2017-12 Issue:23 Volume:27 Page:5179-5184
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Tarr James C.,Wood Michael R.,Noetzel Meredith J.,Melancon Bruce J.,Lamsal Atin,Luscombe Vincent B.,Rodriguez Alice L.,Byers Frank W.,Chang Sichen,Cho Hyekyung P.,Engers Darren W.,Jones Carrie K.,Niswender Colleen M.,Wood Michael W.,Brandon Nicholas J.,Duggan Mark E.,Conn P. Jeffrey,Bridges Thomas M.,Lindsley Craig W.

Funder

NIH

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference30 articles.

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