Discovery of a potent, selective and orally active canine COX-2 inhibitor, 2-(3-difluoromethyl-5-phenyl-pyrazol-1-yl)-5-methanesulfonyl-pyridine-Reference-Cited by-同舟云学术

Discovery of a potent, selective and orally active canine COX-2 inhibitor, 2-(3-difluoromethyl-5-phenyl-pyrazol-1-yl)-5-methanesulfonyl-pyridine

Published:2004-01 Issue:1 Volume:14 Page:95-98
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Li Jin,DeMello Kristin M.Lundy,Cheng Henry,Sakya Subas M.,Bronk Brian S.,Rafka Robert J.,Jaynes Burton H.,Ziegler Carl B.,Kilroy Carolyn,Mann Donald W.,Nimz Eric L.,Lynch Michael P.,Haven Michelle L.,Kolosko Nicole L.,Minich Martha L.,Li Chao,Dutra Jason K.,Rast Bryson,Crosson Rhonda M.,Morton Barry J.,Kirk Glen W.,Callaghan Kathleen M.,Koss David A.,Shavnya Andrei,Lund Lisa A.,Seibel Scott B.,Petras Carol F.,Silvia Annette

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference20 articles.

1. Recently reported inhibitors of cyclooxygenase-2

2. Prostaglandin endoperoxide synthases-1 and -2

3. Chapter 21. Selective Cyclooxygenase-2 Inhibitors

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