Design and synthesis of a novel series of 4-heteroarylamino-1′-azaspiro[oxazole-5,3′-bicyclo[2.2.2]octanes as α7 nicotinic receptor agonists 2. Development of 4-heteroaryl SAR-Reference-Cited by-同舟云学术

Design and synthesis of a novel series of 4-heteroarylamino-1′-azaspiro[oxazole-5,3′-bicyclo[2.2.2]octanes as α7 nicotinic receptor agonists 2. Development of 4-heteroaryl SAR

Published:2017-03 Issue:5 Volume:27 Page:1261-1266
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Iwuagwu Christiana,King Dalton,McDonald Ivar M.,Cook James,Zusi F. Christopher,Hill Matthew D.,Mate Robert A.,Fang Haiquan,Knox Ronald,Gallagher Lizbeth,Post-Munson Amy Easton Debra,Miller Regina,Benitex Yulia,Siuciak Judy,Lodge Nicholas,Zaczek Robert,Morgan Daniel,Bristow Linda,Macor John E.,Olson Richard E.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference40 articles.

1. Longitudinal studies of cognition and functional outcome in schizophrenia: implications for MATRICS

2. Evaluating the role of the alpha-7 nicotinic acetylcholine receptor in the pathophysiology and treatment of schizophrenia

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