Sulfonylureido thiazoles as fructose-1,6-bisphosphatase inhibitors for the treatment of Type-2 diabetes-Reference-Cited by-同舟云学术

Sulfonylureido thiazoles as fructose-1,6-bisphosphatase inhibitors for the treatment of Type-2 diabetes

Published:2010-01 Issue:2 Volume:20 Page:594-599
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Kitas Eric,Mohr Peter,Kuhn Bernd,Hebeisen Paul,Wessel Hans Peter,Haap Wolfgang,Ruf Armin,Benz Jörg,Joseph Catherine,Huber Walter,Sanchez Ruben Alvarez,Paehler Axel,Benardeau Agnes,Gubler Marcel,Schott Brigitte,Tozzo Effie

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference13 articles.

1. The Triumvirate: β-Cell, Muscle, Liver: A Collusion Responsible for NIDDM

2. Increased rate of gluconeogenesis in type II diabetes mellitus. A 13C nuclear magnetic resonance study.

3. Stereoselective synthesis and biological activity of .beta.- and .alpha.-D-arabinose 1,5-diphosphate: analogs of a potent metabolic regulator

4. Anilinoquinazoline Inhibitors of Fructose 1,6-Bisphosphatase Bind at a Novel Allosteric Site: Synthesis, In Vitro Characterization, and X-ray Crystallography

5. MB06322 (CS-917): A potent and selective inhibitor of fructose 1,6-bisphosphatase for controlling gluconeogenesis in type 2 diabetes

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4. Development of disulfide-derived fructose-1,6-bisphosphatase (FBPase) covalent inhibitors for the treatment of type 2 diabetes;European Journal of Medicinal Chemistry;2020-10

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