N-Benzyl-1-heteroaryl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamides as inhibitors of co-activator associated arginine methyltransferase 1 (CARM1)-Reference-Cited by-同舟云学术

N-Benzyl-1-heteroaryl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamides as inhibitors of co-activator associated arginine methyltransferase 1 (CARM1)

Published:2009-02 Issue:4 Volume:19 Page:1218-1223
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Allan Martin,Manku Sukhdev,Therrien Eric,Nguyen Natalie,Styhler Sylvia,Robert Marie-France,Goulet Anne-Christine,Petschner Andrea J.,Rahil Gabi,Robert MacLeod A.,Déziel Robert,Besterman Jeffrey M.,Nguyen Hannah,Wahhab Amal

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference45 articles.

1. State of the Arg

2. Arginine Methylation

3. Protein arginine methyltransferases: Evolution and assessment of their pharmacological and therapeutic potential

4. RNA and Protein Interactions Modulated by Protein Arginine Methylation

5. Transcription regulation by histone methylation: interplay between different covalent modifications of the core histone tails

Cited by 82 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Prodrug Approach to Exploit (S)‐Alanine Amide as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors;ChemMedChem;2024-06-25

2. Overview of the development of protein arginine methyltransferase modulators: Achievements and future directions;European Journal of Medicinal Chemistry;2024-03

3. Trifluoromethyl‐β‐dicarbonyls as Versatile Synthons in Synthesis of Heterocycles;Chemistry – A European Journal;2024-01-04

4. Constitutional adaptation to pK_a modulation by remote ester hydrolysis;Chemical Science;2024

5. Development of selective class I protein arginine methyltransferase inhibitors through fragment-based drug design approach;European Journal of Medicinal Chemistry;2023-11