Synthesis and SAR of heterocyclic carboxylic acid isosteres based on 2-biarylethylimidazole as bombesin receptor subtype-3 (BRS-3) agonists for the treatment of obesity-Reference-Cited by-同舟云学术

Synthesis and SAR of heterocyclic carboxylic acid isosteres based on 2-biarylethylimidazole as bombesin receptor subtype-3 (BRS-3) agonists for the treatment of obesity

Published:2010-05 Issue:9 Volume:20 Page:2912-2915
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Hadden Mark,Goodman Allan,Guo Cheng,Guzzo Peter R.,Henderson Alan J.,Pattamana Kevin,Ruenz Megan,Sargent Bruce J.,Swenson Brian,Yet Larry,Liu Jian,He Shuwen,Sebhat Iyassu K.,Lin Linus S.,Tamvakopoulos Constantin,Peng Qianping,Kan Yanqing,Palyha Oksana,Kelly Theresa M.,Guan Xiao-Ming,Metzger Joseph M.,Reitman Marc L.,Nargund Ravi P.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference15 articles.

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2. Prevalence of Obesity, Diabetes, and Obesity-Related Health Risk Factors, 2001

3. Orlistat

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