Lead optimization of purine based orally bioavailable Mps1 (TTK) inhibitors-Reference-Cited by-同舟云学术

Lead optimization of purine based orally bioavailable Mps1 (TTK) inhibitors

Published:2012-07 Issue:13 Volume:22 Page:4377-4385
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Vijay Kumar D.,Hoarau Christophe,Bursavich Matthew,Slattum Paul,Gerrish David,Yager Kraig,Saunders Michael,Shenderovich Mark,Roth Bruce L.,McKinnon Rena,Chan Ashley,Cimbora Daniel M.,Bradford Chad,Reeves Leslie,Patton Scott,Papac Damon I.,Williams Brandi L.,Carlson Robert O.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference16 articles.

1. The spindle-assembly checkpoint in space and time

2. Human MPS1 Kinase Is Required for Mitotic Arrest Induced by the Loss of CENP-E from Kinetochores

3. Physiological Relevance of Cell Cycle Kinases

4. Targeting Cell Cycle Kinases for Cancer Therapy

5. Cell cycle kinases in cancer

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