7-(Pyrazol-4-yl)-3H-imidazo[4,5-b]pyridine-based derivatives for kinase inhibition: Co-crystallisation studies with Aurora-A reveal distinct differences in the orientation of the pyrazole N1-substituent-Reference-Cited by-同舟云学术

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7-(Pyrazol-4-yl)-3H-imidazo[4,5-b]pyridine-based derivatives for kinase inhibition: Co-crystallisation studies with Aurora-A reveal distinct differences in the orientation of the pyrazole N1-substituent

Published:2015-10 Issue:19 Volume:25 Page:4203-4209
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Bavetsias Vassilios,Pérez-Fuertes Yolanda,McIntyre Patrick J.,Atrash Butrus,Kosmopoulou Magda,O’Fee Lisa,Burke Rosemary,Sun Chongbo,Faisal Amir,Bush Katherine,Avery Sian,Henley Alan,Raynaud Florence I.,Linardopoulos Spiros,Bayliss Richard,Blagg Julian

Funder

CRUK

Breakthrough Breast Cancer Project

MRC CASE

NHS

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference20 articles.

1. Discovery and Development of Aurora Kinase Inhibitors as Anticancer Agents

2. Update on aurora kinase targeted therapeutics in oncology

3. Aurora kinase inhibitors: Progress towards the clinic

4. Aurora Kinases as Anticancer Drug Targets

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1. Imidazo[4,5-b]pyridine derived tubulin polymerization inhibitors: Design, synthesis, biological activity in vitro and computational analysis;Bioorganic Chemistry;2022-10

2. Evaluation of Substituted Pyrazole-Based Kinase Inhibitors in One Decade (2011–2020): Current Status and Future Prospects;Molecules;2022-01-05

3. Recent Progress in Anticancer Agents Incorporating Pyrazole Scaffold;Mini-Reviews in Medicinal Chemistry;2022-01

4. Bicyclic 5-6 Systems: Three Heteroatoms 2:1;Comprehensive Heterocyclic Chemistry IV;2022

5. Novel amino substituted tetracyclic imidazo[4,5-b]pyridine derivatives: Design, synthesis, antiproliferative activity and DNA/RNA binding study;European Journal of Medicinal Chemistry;2021-05

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