One-pot synthesis of novel tert-butyl-4-substituted phenyl-1H-1,2,3-triazolo piperazine/piperidine carboxylates, potential GPR119 agonists-Reference-Cited by-同舟云学术

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One-pot synthesis of novel tert-butyl-4-substituted phenyl-1H-1,2,3-triazolo piperazine/piperidine carboxylates, potential GPR119 agonists

Published:2019-12 Issue:23 Volume:29 Page:126707
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Bashetti Nagaraju,Shanmukha Kumar J.V.,Seelam Naresh Varma,Prasanna B.,Mintz Akiva,Damuka Naresh,Devanathan Sriram,Solingapuram Sai Kiran Kumar

Funder

Wake Forest School of Medicine

CTSA

ADRC

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference20 articles.

1. Pharmacological significance of triazole scaffold;Kharb;J Enzym Inhib Med Chem,2011

2. Synthesis and in vitro characterization of 1-(4-Aminofurazan-3-yl)-5-dialkylaminomethyl-1H-[1,2,3]triazole-4-carboxylic acid derivatives. A new class of selective GSK-3 inhibitors;Olesen;J Med Chem,2003

3. GABA receptors on the somatic muscle cells of the parasitic nematode, Ascaris suum: stereoselectivity indicates similarity to a GABAA-type agonist recognition site;Holden-Dye;Br J Pharmacol,1989

4. Studies on specific inhibition of benzodiazepine receptor binding by some C-benzoyl-1,2,3-triazole derivatives;Biagi;J Pharm Sci,1993

5. Bioisosteres of arecoline: 1,2,3,6-tetrahydro-5-pyridyl-substituted and 3-Piperidyl-substituted derivatives of tetrazoles and 1,2,3-triazoles. synthesis and muscarinic activity;Moltzen;J Med Chem,1994

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1. First GPR119 PET Imaging Ligand: Synthesis, Radiochemistry, and Preliminary Evaluations;Journal of Medicinal Chemistry;2023-06-14

2. GPR119 agonists: Novel therapeutic agents for type 2 diabetes mellitus;Bioorganic Chemistry;2021-08

3. Role of the G protein-coupled receptors GPR84 and GPR119 in the central regulation of food intake in rainbow trout;Journal of Experimental Biology;2021-06-11

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