Preparation and optimization of pyrazolo[1,5- a ]pyrimidines as new potent PDE4 inhibitors-Reference-Cited by-同舟云学术

Preparation and optimization of pyrazolo[1,5- a ]pyrimidines as new potent PDE4 inhibitors

Published:2016-01 Issue:2 Volume:26 Page:454-459
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Le Roux Jacques,Leriche Caroline,Chamiot-Clerc Philippe,Feutrill John,Halley Frank,Papin David,Derimay Nathalie,Mugler Christelle,Grépin Claudine,Schio Laurent

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference26 articles.

1. Primary sequence of cyclic nucleotide phosphodiesterase isozymes and the design of selective inhibitors

2. The Antidepressant and Antiinflammatory Effects of Rolipram in the Central Nervous System

3. PDE4 inhibitors 1998

4. Update on the therapeutic potential of PDE4 inhibitors

5. Inhibitors of PDE4: a review of recent patent literature

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