Discovery of the imidazo[1,5-a][1,2,4]-triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABAA α5 inverse agonist series-Reference-Cited by-同舟云学术

Discovery of the imidazo[1,5-a][1,2,4]-triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABAA α5 inverse agonist series

Published:2009-10 Issue:19 Volume:19 Page:5746-5752
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Achermann Guido,Ballard Theresa M.,Blasco Francesca,Broutin Pierre-Emmanuel,Büttelmann Bernd,Fischer Holger,Graf Martin,Hernandez Maria-Clemencia,Hilty Peter,Knoflach Frédéric,Koblet Andreas,Knust Henner,Kurt Anke,Martin James R.,Masciadri Raffaello,Porter Richard H.P.,Stadler Heinz,Thomas Andrew W.,Trube Gerhard,Wichmann Jürgen

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference50 articles.

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