Discovery of a potent and selective small molecule hGPR91 antagonist-Reference-Cited by-同舟云学术

Discovery of a potent and selective small molecule hGPR91 antagonist

Published:2011-06 Issue:12 Volume:21 Page:3596-3602
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Bhuniya Debnath,Umrani Dhananjay,Dave Bhavesh,Salunke Deepak,Kukreja Gagan,Gundu Jayasagar,Naykodi Minakshi,Shaikh Nadim S.,Shitole Prasad,Kurhade Santosh,De Siddhartha,Majumdar Sreemita,Reddy Srinivasa B.,Tambe Suhas,Shejul Yogesh,Chugh Anita,Palle Venkata P.,Mookhtiar Kasim A.,Cully Doris,Vacca Joseph,Chakravarty Prasun K.,Nargund Ravi P.,Wright Samuel D.,Graziano Michael P.,Singh Sheo B.,Roy Sophie,Cai Tian-Quan

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference26 articles.

1. Citric acid cycle intermediates as ligands for orphan G-protein-coupled receptors

2. The fate of P2Y-related orphan receptors: GPR80/99 and GPR91 are receptors of dicarboxylic acids

3. Anatomical Profiling of G Protein-Coupled Receptor Expression

4. The role of the GPR91 ligand succinate in hematopoiesis

5. The succinate receptor GPR91 in neurons has a major role in retinal angiogenesis

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