Discovery of MK-1439, an orally bioavailable non-nucleoside reverse transcriptase inhibitor potent against a wide range of resistant mutant HIV viruses-Reference-Cited by-同舟云学术

Discovery of MK-1439, an orally bioavailable non-nucleoside reverse transcriptase inhibitor potent against a wide range of resistant mutant HIV viruses

Published:2014-02 Issue:3 Volume:24 Page:917-922
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Côté Bernard,Burch Jason D.,Asante-Appiah Ernest,Bayly Chris,Bédard Leanne,Blouin Marc,Campeau Louis-Charles,Cauchon Elizabeth,Chan Manuel,Chefson Amandine,Coulombe Nathalie,Cromlish Wanda,Debnath Smita,Deschênes Denis,Dupont-Gaudet Kristina,Falgueyret Jean-Pierre,Forget Robert,Gagné Sébastien,Gauvreau Danny,Girardin Melina,Guiral Sébastien,Langlois Eric,Li Chun Sing,Nguyen Natalie,Papp Rob,Plamondon Serge,Roy Amélie,Roy Stéphanie,Seliniotakis Ria,St-Onge Miguel,Ouellet Stéphane,Tawa Paul,Truchon Jean-François,Vacca Joe,Wrona Marc,Yan Youwei,Ducharme Yves

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference17 articles.

1. Progress and Problems in the Fight against AIDS

2. Treatment for Adult HIV Infection

3. An Overview of Mitochondrial Toxicity of Nucleoside Reverse Transcriptase Inhibitors Associated with HIV Therapy

4. Conformational Changes in HIV-1 Reverse Transcriptase Induced by Nonnucleoside Reverse Transcriptase Inhibitor Binding

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