Pyrrolidine-constrained phenethylamines: The design of potent, selective, and pharmacologically efficacious dipeptidyl peptidase IV (DPP4) inhibitors from a lead-like screening hit-Reference-Cited by-同舟云学术

Pyrrolidine-constrained phenethylamines: The design of potent, selective, and pharmacologically efficacious dipeptidyl peptidase IV (DPP4) inhibitors from a lead-like screening hit

Published:2007-04 Issue:7 Volume:17 Page:2005-2012
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Backes Bradley J.,Longenecker Kenton,Hamilton Gregory L.,Stewart Kent,Lai Chunqiu,Kopecka Hana,von Geldern Thomas W.,Madar David J.,Pei Zhonghua,Lubben Thomas H.,Zinker Bradley A.,Tian Zhenping,Ballaron Stephen J.,Stashko Michael A.,Mika Amanda K.,Beno David W.A.,Kempf-Grote Anita J.,Black-Schaefer Candace,Sham Hing L.,Trevillyan James M.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference35 articles.

1. Effect of 6-week course of glucagon-like peptide 1 on glycaemic control, insulin sensitivity, and β-cell function in type 2 diabetes: a parallel-group study

2. Glucagonlike peptide 1: A newly discovered gastrointestinal hormone

3. Glucagon-like peptides

4. Glucagon-like peptide-1: A basis for new approaches to the management of diabetes

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