Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 1: Discovery and SAR study of 4-pyrazolylpiperidine side chains-Reference-Cited by-同舟云学术

Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 1: Discovery and SAR study of 4-pyrazolylpiperidine side chains

Published:2004-02 Issue:4 Volume:14 Page:935-939
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Shen Dong-Ming,Shu Min,Mills Sander G.,Chapman Kevin T.,Malkowitz Lorraine,Springer Martin S.,Gould Sandra L.,DeMartino Julie A.,Siciliano Salvatore J.,Kwei Gloria Y.,Carella Anthony,Carver Gwen,Holmes Karen,Schleif William A.,Danzeisen Renee,Hazuda Daria,Kessler Joseph,Lineberger Janet,Miller Michael D.,Emini Emilio A.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference21 articles.

1. The chemokine/chemokine-receptor family: potential and progress for therapeutic intervention

2. Co-receptor use by HIV and inhibition of HIV infection by chemokine receptor ligands

3. Homozygous Defect in HIV-1 Coreceptor Accounts for Resistance of Some Multiply-Exposed Individuals to HIV-1 Infection

4. HIV-1 entry – an expanding portal for drug discovery

5. Chemokine Receptor Antagonists

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