3D-QSAR and 3D-QSSR models of negative allosteric modulators facilitate the design of a novel selective antagonist of human α4β2 neuronal nicotinic acetylcholine receptors-Reference-Cited by-同舟云学术

3D-QSAR and 3D-QSSR models of negative allosteric modulators facilitate the design of a novel selective antagonist of human α4β2 neuronal nicotinic acetylcholine receptors

Published:2012-02 Issue:4 Volume:22 Page:1797-1813
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Henderson Brandon J.,Orac Crina M.,Maciagiewicz Iwona,Bergmeier Stephen C.,McKay Dennis B.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference23 articles.

1. Brain nicotinic acetylcholine receptors: native subtypes and their relevance

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3. Nicotine Activation of α4* Receptors: Sufficient for Reward, Tolerance, and Sensitization

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