Dihydropyrrolopyrazol-6-one MCHR1 antagonists for the treatment of obesity: Insights on in vivo efficacy from a novel FLIPR assay setup-Reference-Cited by-同舟云学术

Dihydropyrrolopyrazol-6-one MCHR1 antagonists for the treatment of obesity: Insights on in vivo efficacy from a novel FLIPR assay setup

Published:2015-07 Issue:14 Volume:25 Page:2793-2799
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Devasthale Pratik,Wang Wei,Hernandez Andres S.,Moore Fang,Renduchintala Kishore,Sridhar Radhakrishnan,Pelleymounter Mary Ann,Longhi Daniel,Huang Ning,Flynn Neil,Azzara Anthony V.,Rohrbach Kenneth,Devenny James,Rooney Suzanne,Thomas Michael,Glick Susan,Godonis Helen,Harvey Susan,Cullen Mary Jane,Zhang Hongwei,Caporuscio Christian,Stetsko Paul,Grubb Mary,Huang Christine,Zhang Lisa,Freeden Chris,Li Yi-Xin,Murphy Brian J.,Robl Jeffrey A.,Washburn William N.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference14 articles.

1. World Health Organization Global Health Observatory (GHO) website http://www.who.int/mediacentre/factsheets/fs311/en/ (updated Aug 2014).

2. Antiobesity Pharmacotherapy: New Drugs and Emerging Targets

3. Novel MCH1receptor antagonists: a patent review

4. Recent Patents on Novel MCH1 Receptor Antagonists as Potential Anti-Obesity Drugs

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