Discovery of boronic acid-based potent activators of tumor pyruvate kinase M2 and development of gastroretentive nanoformulation for oral dosing-Reference-Cited by-同舟云学术

Discovery of boronic acid-based potent activators of tumor pyruvate kinase M2 and development of gastroretentive nanoformulation for oral dosing

Published:2021-06 Issue: Volume:42 Page:128062
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Patle Rajkumar,Shinde Shital,Patel Sagarkumar,Maheshwari Rahul,Jariyal Heena,Srivastava Akshay,Chauhan Neelam,Globisch Christoph,Jain Alok,Tekade Rakesh K.,Shard Amit

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference69 articles.

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4. Dual roles of PKM2 in cancer metabolism;Wu;Acta Biochim Biophys Sin,2013

5. Tumor pyruvate kinase M2: a promising molecular target of gastrointestinal cancer;Guo;Chinese J Cancer Res,2018

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