Novel 1-(prop-2-yn-1-ylamino)-2,3-dihydro-1H-indene-4-thiol derivatives as potent selective human monoamine oxidase B inhibitors: Design, SAR development, and biological evaluation-Reference-Cited by-同舟云学术

Novel 1-(prop-2-yn-1-ylamino)-2,3-dihydro-1H-indene-4-thiol derivatives as potent selective human monoamine oxidase B inhibitors: Design, SAR development, and biological evaluation

Published:2021-07 Issue: Volume:43 Page:128051
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Kong Haiyan,Meng Xianshe,Hou Rui,Yang Xiaoxiao,Han Jihong,Xie Zhouling,Duan Yajun,Liao Chenzhong^ORCID

Funder

National Natural Science Foundation of China

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference20 articles.

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2. Regulation of MAO-A and MAO-B gene expression;Shih;Curr Med Chem,2004

3. Structure and mechanism of monoamine oxidase;Edmondson;Curr Med Chem.,2004

4. Structural insights into the mechanism of amine oxidation by monoamine oxidases A and B;Edmondson;Arch Biochem Biophys,2007

5. Use of monoamine oxidase inhibitors in chronic neurodegeneration;Riederer;Expert Opin Drug Met,2017

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1. Organic compounds based on 1-(prop-2-yn-1-ylamino)-2,3-dihydro-1H-indene-4-thiol as selective human monoamine oxidase B inhibitors. Quantitative analysis of structure-activity relationships and in-silico investigations;MOROC J CHEM;2023

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