Design, synthesis, and biological evaluation of monopyrrolinone-based HIV-1 protease inhibitors possessing augmented P2′ side chains-Reference-Cited by-同舟云学术

Design, synthesis, and biological evaluation of monopyrrolinone-based HIV-1 protease inhibitors possessing augmented P2′ side chains

Published:2006-02 Issue:4 Volume:16 Page:859-863
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Smith Amos B.,Charnley Adam K.,Harada Hironori,Beiger Jason J.,Cantin Louis-David,Kenesky Craig S.,Hirschmann Ralph,Munshi Sanjeev,Olsen David B.,Stahlhut Mark W.,Schleif William A.,Kuo Lawrence C.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference27 articles.

1. New Anti-HIV Agents in Preclinical or Clinical Development

2. New Approaches toward Anti-HIV Chemotherapy

3. (b) Condra, J. H.; Vacca, J. P. HIV-1 protease inhibitors. In The Human Immunodeficiency Virus: Biology, Immunology, and Therapy; Emini E. A. Ed.; Princeton University Press, Princeton, NJ, 2002; pp 172–222.

4. Protease Inhibitors: Current Status and Future Prospects

5. Design, synthesis, and crystal structure of a pyrrolinone-based peptidomimetic possessing the conformation of a .beta.-strand: potential application to the design of novel inhibitors of proteolytic enzymes

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