Pharmacokinetics and metabolism studies on (3-tert-butyl-7-(5-methylisoxazol-3-yl)-2-(1-methyl-1H-1,2,4-triazol-5-ylmethoxy) pyrazolo[1,5-d][1,2,4]triazine, a functionally selective GABAA α5 inverse agonist for cognitive dysfunction-Reference-Cited by-同舟云学术

Pharmacokinetics and metabolism studies on (3-tert-butyl-7-(5-methylisoxazol-3-yl)-2-(1-methyl-1H-1,2,4-triazol-5-ylmethoxy) pyrazolo[1,5-d][1,2,4]triazine, a functionally selective GABAA α5 inverse agonist for cognitive dysfunction

Published:2006-02 Issue:4 Volume:16 Page:872-875
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Jones Philip,Atack John R.,Braun Matthew P.,Cato Brian P.,Chambers Mark S.,O’Connor Desmond,Cook Susan M.,Hobbs Sarah C.,Maxey Robert,Szekeres Helen J.,Szeto Nicola,Wafford Keith A.,MacLeod Angus M.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference18 articles.

1. theta , a novel gamma -aminobutyric acid type A receptor subunit

2. Which GABAA-receptor subtypes really occur in the brain?

3. SEVERE ANXIETY INDUCED BY FG 7142, A β-CARBOLINE LIGAND FOR BENZODIAZEPINE RECEPTORS

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