Design, synthesis and structure–activity relationships of (indo-3-yl) heterocyclic derivatives as agonists of the CB1 receptor. Discovery of a clinical candidate-Reference-Cited by-同舟云学术

Design, synthesis and structure–activity relationships of (indo-3-yl) heterocyclic derivatives as agonists of the CB1 receptor. Discovery of a clinical candidate

Published:2011-04 Issue:8 Volume:21 Page:2541-2546
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Ratcliffe Paul,Adam Julia M.,Baker James,Bursi Roberta,Campbell Robert,Clark John K.,Cottney Jean E.,Deehan Maureen,Easson Anna-Marie,Ecker Daniel,Edwards Darren,Epemolu Ola,Evans Louise,Fields Ruth,Francis Stuart,Harradine Paul,Jeremiah Fiona,Kiyoi Takao,McArthur Duncan,Morrison Angus,Passier Paul,Pick Jack,Schnabel Peter G.,Schulz Jurgen,Steinbrede Heinz,Walker Glenn,Westwood Paul,Wishart Grant,Haes Joanna Udo de

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference14 articles.

1. Recent Developments in the Medicinal Chemistry of Cannabimimetic Indoles, Pyrroles and Indenes

2. CB1 Cannabinoid Antagonists: Structure-Activity Relationships and Potential Therapeutic Applications

3. The endocannabinoid system, eating behavior and energy homeostasis: The end or a new beginning?

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