Design and evaluation of 3,6-di(hetero)aryl imidazo[1,2-a]pyrazines as inhibitors of checkpoint and other kinases-Reference-Cited by-同舟云学术

Design and evaluation of 3,6-di(hetero)aryl imidazo[1,2-a]pyrazines as inhibitors of checkpoint and other kinases

Published:2010-07 Issue:14 Volume:20 Page:4045-4049
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Matthews Thomas P.,McHardy Tatiana,Klair Suki,Boxall Kathy,Fisher Martin,Cherry Michael,Allen Charlotte E.,Addison Glynn J.,Ellard John,Aherne G. Wynne,Westwood Isaac M.,Montfort Rob van,Garrett Michelle D.,Reader John C.,Collins Ian

Funder

Cancer Research UK [CUK]

The Institute of Cancer Research

NHS

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference24 articles.

1. Protein kinases — the major drug targets of the twenty-first century?

2. Heteroaromatic Rings of the Future

3. Breaching the DNA damage checkpoint via PF-00477736, a novel small-molecule inhibitor of checkpoint kinase 1

4. DNA Damage Detection and Repair Pathways—Recent Advances with Inhibitors of Checkpoint Kinases in Cancer Therapy

5. G2 checkpoint abrogation and checkpoint kinase-1 targeting in the treatment of cancer

Cited by 27 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Novel imidazolone derivatives as potential dual inhibitors of checkpoint kinases 1 and 2: Design, synthesis, cytotoxicity evaluation, and mechanistic insights;Bioorganic Chemistry;2024-08

2. The Discovery of Checkpoint Kinase 1 Inhibitors: From Fragments to Clinical Candidate;The Handbook of Medicinal Chemistry;2023-02-03

3. Recent Developments in the Synthesis of Indole‐Pyrazole Hybrids;ChemistrySelect;2022-06

4. A Diverse Benchmark Based on 3D Matched Molecular Pairs for Validating Scoring Functions;ACS Omega;2018-05-28

5. An Update on Direct C–H Bond Functionalization of Nitrogen-Containing Fused Heterocycles;Synthesis;2017-08-25