Design and SAR of selective T-type calcium channel antagonists containing a biaryl sulfonamide core-Reference-Cited by-同舟云学术

Design and SAR of selective T-type calcium channel antagonists containing a biaryl sulfonamide core

Published:2008-01 Issue:2 Volume:18 Page:474-478
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Hangeland Jon J.,Cheney Daniel L.,Friends Todd J.,Swartz Stephen,Levesque Paul C.,Rich Adam J.,Sun Lucy,Bridal Terry R.,Adam Leonard P.,Normandin Diane E.,Murugesan Natesan,Ewing William R.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference27 articles.

1. Structure and Regulation of Voltage-Gated Ca2+ Channels

2. Molecular Physiology of Low-Voltage-Activated T-type Calcium Channels

3. Discovery and main pharmacological properties of mibefradil (Ro 40-5967), the first selective T-type calcium channel blocker

4. Efonidipine Hydrochloride: A New Calcium Antagonist

5. Efonidipine Hydrochloride: A Dual Blocker of L- and T-Type Ca2+ Channels

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