Synthesis and SAR of analogs of the M1 allosteric agonist TBPB. Part II: Amides, sulfonamides and ureas—The effect of capping the distal basic piperidine nitrogen-Reference-Cited by-同舟云学术

Synthesis and SAR of analogs of the M1 allosteric agonist TBPB. Part II: Amides, sulfonamides and ureas—The effect of capping the distal basic piperidine nitrogen

Published:2008-10 Issue:20 Volume:18 Page:5443-5447
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Miller Nicole R.,Daniels R. Nathan,Bridges Thomas M.,Brady Ashley E.,Conn P. Jeffrey,Lindsley Craig W.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference15 articles.

1. Identification of a Family of Muscarinic Acetylcholine Receptor Genes

2. Cloning and expression of the human and rat m5 muscarinic acetylcholine receptor genes

3. Therapeutic Opportunities for Muscarinic Receptors in the Central Nervous System

4. Muscarinic receptor ligands and their therapeutic potential

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