Identification of novel PI3K inhibitors through a scaffold hopping strategy-Reference-Cited by-同舟云学术

Identification of novel PI3K inhibitors through a scaffold hopping strategy

Published:2017-11 Issue:21 Volume:27 Page:4794-4799
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Martínez González Sonia,Hernández Ana Isabel,Álvarez Rosa María,Rodríguez Antonio,Ramos-Lima Francisco,Bischoff James R.,Albarrán María Isabel,Cebriá Antonio,Hernández-Encinas Elena,García-Arocha Jennifer,Cebrián David,Blanco-Aparicio Carmen,Pastor Joaquín

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference23 articles.

1. Bioisosteres and Scaffold Hopping in Medicinal Chemistry

2. Classification of scaffold-hopping approaches

3. Konkol LC, Senter TJ, Lindsley CW. Methods and Principles in Medicinal Chemistry 2014, 58, (Scaffold Hopping in Medicinal Chemistry), 247–257.

4. Scaffold-Hopping: How Far Can You Jump?

5. Kinase Patent Space Visualization Using Chemical Replacements

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