Structural optimization and biological evaluation of 1,5-disubstituted pyrazole-3-carboxamines as potent inhibitors of human 5-lipoxygenase-Reference-Cited by-同舟云学术

Structural optimization and biological evaluation of 1,5-disubstituted pyrazole-3-carboxamines as potent inhibitors of human 5-lipoxygenase

Published:2016-01 Issue:1 Volume:6 Page:32-45
ISSN:2211-3835
Container-title:Acta Pharmaceutica Sinica B
language:en
Short-container-title:Acta Pharmaceutica Sinica B

Author:

Zhou Yu,Liu Jun,Zheng Mingyue,Zheng Shuli,Jiang Chunyi,Zhou Xiaomei,Zhang Dong,Zhao Jihui,Ye Deju,Zheng Mingfang,Jiang Hualiang,Liu Dongxiang,Cheng Jian,Liu Hong

Funder

National Natural Science Foundation of China

Major Project of Chinese National Programs for Fundamental Research and Development

National High Technology Research and Development Program of China

National Basic Research Program of China

National S&T Major Projects

Publisher

Elsevier BV

Subject

General Pharmacology, Toxicology and Pharmaceutics

Reference33 articles.

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3. Recent advances in the search for novel 5-lipoxygenase inhibitors;Steinhilber;Basic Clin Pharmacol Toxicol,2014

4. Leukotrienes, antileukotrienes and asthma;Montuschi;Mini Rev Med Chem,2008

5. 5-Lipoxygenase inhibitors: a review of recent patents (2010–2012);Hofmann;Expert Opin Ther Pat,2013

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