Discovery of L-740,515, a potent thienopyridine cysLT1 receptor (LTD4 receptor) antagonist-Reference-Cited by-同舟云学术

Discovery of L-740,515, a potent thienopyridine cysLT1 receptor (LTD4 receptor) antagonist

Published:1995-11 Issue:21 Volume:5 Page:2551-2556
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Labelle M.,Gareau Y.,Dufresne C.,Lau C.K.,Belley M.,Jones T.R.,Leblanc Y.,McAuliffe M.,McFarlane C.S.,Metters K.M.,Ouimet N.,Perrier H.,Rochette C.,Sawyer N.,Slipetz D.,Xiang Y.B.,Wang Z.,Pickett C.B.,Ford-Hutchinson A.W.,Young R.N.,Zamboni R.J.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference22 articles.

1. 677 The therapeutic effects of MK-571, a potent and selective leukotriene (LT) D receptor antagonist, in patients with chronic asthma

2. Lung function improvement in asthma with a cysteinylleukotriene receptor antagonist

3. The discovery of a new structural class of potent orally active leukotriene D4 antagonists

4. The discovery of L-699,392, a novel potent and orally active leukotriene D4 receptor antagonist

5. Enantioselective induction of peroxisomal proliferation in CD-1 mice by leukotriene antagonists

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1. Classification models and SAR analysis on CysLT1 receptor antagonists using machine learning algorithms;Molecular Diversity;2021-02-03

2. ChemInform Abstract: Discovery of L-740,515, a Potent Thienopyridine cysLT1 Receptor (LTD4 Receptor) Antagonist.;ChemInform;2010-08-12

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4. Comparison between two classes of selective EP3 antagonists and their biological activities;Bioorganic & Medicinal Chemistry Letters;2006-11

5. 5 Discovery of Montelukast: a Once-a-Day Oral Antagonist of Leukotriene D4 for the Treatment of Chronic Asthma;Progress in Medicinal Chemistry;2001