Potent fluoromethyl ketone inhibitors of recombinant human calpain I-Reference-Cited by-同舟云学术

Potent fluoromethyl ketone inhibitors of recombinant human calpain I

Published:1996-06 Issue:11 Volume:6 Page:1237-1240
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Chatterjee Sankar,Josef Kurt,Wells Gregory,Iqbal Mohamed,Bihovsky Ron,Mallamo John P.,Ator Mark A.,Bozyczko-Coyne Donna,Mallya Satish,Senadhi Shobha,Siman Robert

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference21 articles.

1. Calcium-activated neutral protease (calpain) system: structure, function, and regulation.

2. Calpain inhibition: an overview of its therapeutic potential

3. Cell-penetrating inhibitors of calpain

4. Stereospecific Synthesis of Peptidyl .alpha.-Keto Amides as Inhibitors of Calpain

5. Peptide .alpha.-keto ester, .alpha.-keto amide, and .alpha.-keto acid inhibitors of calpains and other cysteine proteases

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