Evidence for low brain penetration by the H1-receptor antagonist temelastine (SK & F 93944)
Author:
Publisher
Elsevier BV
Subject
Pharmacology
Reference23 articles.
1. Dissociation de deux composants dans le compartement d'investigation de la souris;Boissier;Arch. Int. Pharmacodyn. Ther.,1964
2. Pharmacological studies with SK & F 93944 (temelastine), a novel histamine H1-receptor antagonist with negligible ability to penetrate the central nervous system;Brown;Br. J. Pharmacol.,1986
3. Heterogeneity of histamine H1-receptors: species variations in [3H]mepyramine binding of brain membranes;Chang;J. Neurochem.,1979
4. Antihistamine effect of terfenadine: a new piperidine-type antihistamine;Cheng;Drug Dev. Res.,1982
5. Histamine H1-agonist potentiation of adenosine-stimulated cyclic AMP accumulation in slices of guinea-pig cerebral cortex: comparison of response and binding parameters;Daum;Br. J. Pharmacol.,1982
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1. Serum protein binding of histamine H1-antagonists. A comparative study on the serum protein binding of a sedating ([3H]mepyramine) and a non-sedating H1-antagonist ([3H]loratadine);European Journal of Pharmaceutical Sciences;1996-09
2. Characteristics of the binding of [3H]-mepyramine to intact human U373 MG astrocytoma cells: evidence for histamine-induced H1-receptor internalisation;British Journal of Pharmacology;1995-11
3. Molecular pharmacological aspects of histamine receptors;Pharmacology & Therapeutics;1995-01
4. Pharmacology of the Histaminergic System;Handbook of Experimental Pharmacology;1995
5. Lipophilicity and hydrogen-bonding capacity of H1-antihistaminic agents in relation to their central sedative side-effects;European Journal of Pharmaceutical Sciences;1994-12
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