Design, synthesis and anti-HIV evaluation of 5-alkyl- 6-(benzo[d][1,3]dioxol-5-alkyl)-2-mercaptopyrimidin-4(3H)-ones as potent HIV-1 NNRTIs

Author:

Li Yi-Ming,Luo Rong-Hua,Yang Liu-Meng,Huang Si-Ming,Li Sui-Yuan,Zheng Yu-Gui,Ni Dong-Xuan,Cui Yi-Man,Zhang Xing-Jie,Li Xiao-Li,Zhang Rui-Han,Tang E,Zhang Hong-Bin,Zheng Yong-Tang,He Yan-Ping,Xiao Wei-Lie

Funder

National Natural Science Foundation of China

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference48 articles.

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2. The journey of HIV-1 non-nucleoside reverse transcriptase inhibitors (NNRTIs) from lab to clinic;Namasivayam;J. Med. Chem.,2019

3. Combined approaches for HIV cure;Margolis;Curr. Opin.,2013

4. Current status and challenges of antiretroviral research and therapy;Este;Antivir. Res.,2010

5. D. Finzi, M. Hermankova, T. Pierson, L. M. et al., Identification of a reservoir for HIV-1 in patients on highly active antiretroviral therapy, Science. 278 (1997), 1295-300.

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