Design of iodinated radioligands for SPECT imaging of central human 5-HT4R using a ligand lipophilicity efficiency approach-Reference-Cited by-同舟云学术

Design of iodinated radioligands for SPECT imaging of central human 5-HT4R using a ligand lipophilicity efficiency approach

Published:2020-03 Issue: Volume:96 Page:103582
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Babin Victor,Tournier Benjamin B.,Davis Audrey,Dubost Emmanuelle,Pigrée Gilbert,Lohier Jean-François,Reboul Vincent,Cailly Thomas,Bouillon Jean-Philippe,Millet Philippe,Fabis Frédéric

Funder

European Regional Development Fund

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

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5. A 5-HT receptor in the central nervous system, positively coupled with adenylate cyclase, is antagonized by ICS 205 930;Dumuis;Eur. J. Pharmacol.,1988

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