Identification and development of thiazole leads as COX-2/5-LOX inhibitors through in-vitro and in-vivo biological evaluation for anti-inflammatory activity-Reference-Cited by-同舟云学术

Identification and development of thiazole leads as COX-2/5-LOX inhibitors through in-vitro and in-vivo biological evaluation for anti-inflammatory activity

Published:2020-07 Issue: Volume:100 Page:103882
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Jacob P Jaismy,Manju S.L.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference48 articles.

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3. Safer anti-inflammatory therapy through dual COX-2/5-LOX inhibitors: a structure-based approach;Jacob;Eur. J. Pharm. Sci.,2018

4. Thiazoles and thiazolidinones as COX/LOX inhibitors;Liaras;Molecules,2018

5. Synthesis, biological evaluation, docking study and ulcerogenicity profiling of some novel quinoline-2-carboxamides as dual COXs/LOX inhibitors endowed with anti-inflammatory activity;Abdelrahman;Eur. J. Med. Chem.,2017

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