Design, synthesis and biological evaluation of new series of hexahydroquinoline and fused quinoline derivatives as potent inhibitors of wild-type EGFR and mutant EGFR (L858R and T790M)-Reference-Cited by-同舟云学术

Design, synthesis and biological evaluation of new series of hexahydroquinoline and fused quinoline derivatives as potent inhibitors of wild-type EGFR and mutant EGFR (L858R and T790M)

Published:2020-12 Issue: Volume:105 Page:104274
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Shaheen Mennatallah A.,El-Emam Ali A.,El-Gohary Nadia S.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference88 articles.

1. Estimating the global cancer incidence and mortality in 2018: GLOBOCAN sources and methods;Ferlay;Int. J. Cancer,2019

2. Population-based study of surgical treatment with and without tumour resection in patients with locally recurrent rectal cancer;Westberg;Br. J. Surg.,2019

3. Losartan treatment enhances chemotherapy efficacy and reduces ascites in ovarian cancer models by normalizing the tumor stroma;Zhao;Proc. Natl. Acad. Sci.,2019

4. Development and feasibility of a swallowing intervention package (SiP) for patients receiving radiotherapy treatment for head and neck cancer-the SiP study protocol;Wells;Pilot Feasibility Stud.,2016

5. Untangling the ErbB signalling network;Yarden;Nat. Rev. Mol. Cell Biol.,2001

Cited by 16 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Structural Perspectives in the Development of Novel EGFR Inhibitors for the Treatment of NSCLC;Mini-Reviews in Medicinal Chemistry;2024-10

2. Novel Pyrimidine-5-Carbonitriles as potential apoptotic and antiproliferative agents by dual inhibition of EGFRWT/T790M and PI3k enzymes; Design, Synthesis, biological Evaluation, and docking studies;Bioorganic Chemistry;2024-04

3. Syntheses, characterizations, crystal structures and Hirshfeld surface analyses of methyl 4-[4-(difluoromethoxy)phenyl]-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate, isopropyl 4-[4-(difluoromethoxy)phenyl]-2,6,6-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate and tert-butyl 4-[4-(difluoromethoxy)phenyl]-2,6,6-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate;Acta Crystallographica Section E Crystallographic Communications;2024-02-08

4. Synthesis, biological evaluation and network pharmacology based studies of 1,3,4-oxadiazole bearing azaphenols as anticancer agents;Arabian Journal of Chemistry;2024-01

5. 1,4-Dihydropyridine Derivatives: An Overview of Synthesis Conditions and Biological Tests;Current Organic Chemistry;2023-10